GSK 525762A （Cas No.1260907-17-2)
Product Quick Detail
- Cas No.
- 1260907-17-2
- M.Wt
- 423.9
- Solubility
- DMSO
- Formula
- C22H22ClN5O2
- Purity
- 98%
- Synonyms
- GSK525762A; GSK-525762A; I-BET762; I-BET 762
- Packaging
- Fluorinated Bottles
- Delivery
- 7 Days
Specifications
GSK 525762A is an inhibitor for BET (bromodomain and extra terminal domain) proteins, BRD2, BRD3 and BRD4, binds to the tandem bromodomains of BET with Kd of 50.5-61.3 nM, displaces
a tetra-acetylated H4 peptide prebound to tandem bromodomains of BET with IC50 of 32.5-42.5 nM in FRET analysis. GSK 525762A occupies the acetyl-lysine binding pocket of BET proteins and inhibits
binding of BET proteins to acetylated histones, thus disrupts the formation of the chromatin complexes essential for expression of inflammatory genes.
- Country: China (Mainland)
- Business Type:
- Market:European Union,Americas
- Founded Year:2009
- Address:武汉东湖高新区长城科技园光谷精工D栋402室
- Contact:Rosie Liu
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